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Wyszukujesz frazę "Shah, R. R." wg kryterium: Autor


Tytuł:
Mesomorphic properties of liquid crystalline compounds with central linkage chalconyl ester and laterally substituted bromo group
Autorzy:
Patel, Patel
Patel, R. B.
Shah, R. R.
Powiązania:
https://bibliotekanauki.pl/articles/1191246.pdf
Data publikacji:
2016
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
Nematic; Liquid crystalline; Mesomorphic; Enantiotropic
Smectic
Opis:
To investigate the mesomorphic property of the substitution on mesomorphism, the new series of liquid crystals having the following structures have been synthesized. Presently synthesized series contain thirteen homologue (C1 to C8, C10, C12, C14, C16, C18) in which eleven homologue (C3 to C18) shows both smectic as well as nematic phase during heating and cooling condition in enantiotropic manner, while C2 homologue shows only nematic phase. All the homologues were characterised by elemental analysis and spectroscopic techniques like 1H-NMR and IR analysis. Their liquid crystalline behaviours were measured by polarised optical microscope (POM) and Differencial Scanning Calorimetry (DSC).
Źródło:
World Scientific News; 2016, 54; 202-216
2392-2192
Pojawia się w:
World Scientific News
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
A new mechanism for data visualization with TSK-type preprocessed collaborative fuzzy rule based system
Autorzy:
Prasad, M.
Liu, Y.-T.
Li, D.-L.
Lin, C. -T.
Shah, R. R.
Kaiwartya, O. P.
Powiązania:
https://bibliotekanauki.pl/articles/91743.pdf
Data publikacji:
2017
Wydawca:
Społeczna Akademia Nauk w Łodzi. Polskie Towarzystwo Sieci Neuronowych
Tematy:
fuzzy interference system
collaborative clustering
fuzzy logic
big data
data visualization
Opis:
A novel data knowledge representation with the combination of structure learning ability of preprocessed collaborative fuzzy clustering and fuzzy expert knowledge of TakagiSugeno-Kang type model is presented in this paper. The proposed method divides a huge dataset into two or more subsets of dataset. The subsets of dataset interact with each other through a collaborative mechanism in order to find some similar properties within eachother. The proposed method is useful in dealing with big data issues since it divides a huge dataset into subsets of dataset and finds common features among the subsets. The salient feature of the proposed method is that it uses a small subset of dataset and some common features instead of using the entire dataset and all the features. Before interactions among subsets of the dataset, the proposed method applies a mapping technique for granules of data and centroid of clusters. The proposed method uses information of only half or less/more than the half of the data patterns for the training process, and it provides an accurate and robust model, whereas the other existing methods use the entire information of the data patterns. Simulation results show the proposed method performs better than existing methods on some benchmark problems.
Źródło:
Journal of Artificial Intelligence and Soft Computing Research; 2017, 7, 1; 33-46
2083-2567
2449-6499
Pojawia się w:
Journal of Artificial Intelligence and Soft Computing Research
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
An efficient one-pot multicomponent synthesis and characterization of 5-cyano-1,2,3,4-tetrahydropyrimidine derivatives
Autorzy:
Vaghasiya, R. G.
Shah, V. H.
Powiązania:
https://bibliotekanauki.pl/articles/411702.pdf
Data publikacji:
2015
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
substituted pyrazole-4-carbaldehyde
5-cyano-1,2,3,4-tetrahydropyrimidine derivatives
multi component reaction
non-chromatographic method
Opis:
A series of pyrimidine-5-carbonitrile derivatives was efficiently synthesized via one-pot, multi component reaction (MCRs) of 1,3-bifunctional synthon (ethylcyano acetate), substituted pyrazole-4-carbaldehyde, and thiourea/urea in the presence of basic catalyst. The key advantages of this process are high yields, shorter reaction times, easy work-up, and purification of products by non-chromatographic method.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2015, 40; 51-60
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Synthesis, Characterization and Biological evaluation of 6-substituted-2-(substituted-phenyl)-quinoline derivatives bearing 4-amino-1,2,4-triazole-3-thiol ring at C-4 position
Autorzy:
Vaghasiya, R. G.
Ghodasara, H. B.
Vachharajani, P. R.
Shah, V. H.
Powiązania:
https://bibliotekanauki.pl/articles/412211.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
Quinoline, 4-amino-1,2,4-triazole-3-thiol
therapeutic agents
antimicrobial assai
Opis:
Quinoline derivatives represent one of the most active classes of compounds possesses wide spectrum biodynamic activities and use as potent therapeutic agents. In this research work, a synthesis, characterization and biological evaluation of 6-substituted-2-(substituted-phenyl)-quinoline derivatives bearing 4-amino-1,2,4-triazole-3-thiol ring at C-4 position is described. The synthesis of quinoline derivatives is carried out by the reaction of substituted quinoline-4-carbohydrazides with a mixture of carbon disulphide and potassium hydroxide which further react with hydrazine hydrate to give final compounds. All of these compounds were screened for their in vitro antimicrobial assay against gram (+ve), gram (-ve) bacteria and fungi activity compared with standard drugs viz., Ampicilin, Chloramphenicol, Ciprofloxacin, Norfloxacin, Griseofulvin and Nystatin at different concentrations.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 8; 30-37
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Synthesis, characterization of biologically potent novel chalcones bearing urea, thiourea and acetamide linkages
Autorzy:
Mewada, N. S.
Shah, D. R.
Chikhalia, K. H.
Powiązania:
https://bibliotekanauki.pl/articles/412032.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
Chalcone
urea
thiourea
acetamide
antimicrobial activity and antifungal activity
Opis:
Three series of some novel chalcone based urea, thiourea and acetamide derivatives were designed, synthesized and screened for their antimicrobial and antifungal activities. All the synthesized compounds are first reported. The structures of the compounds were elucidated with the aid of elemental analysis and spectral methods including IR, 1H-NMR spectral data. The prepared compounds were evaluated for antibacterial activity against two Gram-positive bacteria (Staphylococcus aureus, Staphylococcus pyogenus), two Gram-negative bacteria (Pseudomonas aeruginosa, Escherichia coli). The title compounds were also investigated for their antifungal activity using the broth micro dilution method. The bioassay results showed that compounds a few compounds showed good to superior in vitro antibacterial and antifungal activity.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 17, 3; 281-294
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Synthesis, characterization and docking studies of some novel xanthene derivatives
Autorzy:
Bhatt, Aditya H.
Shah, Viral R.
Rawal, Rakesh M.
Powiązania:
https://bibliotekanauki.pl/articles/1075739.pdf
Data publikacji:
2019
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
Antimicrobial activity
Docking studies
Hantzsch synthesis
Xanthene
Opis:
The synthesis of a novel xanthene derivatives bearing dimedone as an excellent precursor has been achieved by applying one pot three component Hantzsch type condensation. The newly synthesized compounds were characterized by spectral and elemental analyses. All synthesized compounds undergo docking studies and biological screening for antimicrobial activity against Gram-positive bacteria, Gram-negative bacteria and fungal species. Among all the tested compounds, it was found that compound 3c, 3d, 3g and 3h revealed better activities against the Gram-positive rather than the Gram-negative bacteria whereas results of docking studies revealed that compounds 3b, 3g and 3i showed best binding affinity towards ATP binding pocket of Human PIM1 kinase receptor through steric favorable and H-bond interactions.
Źródło:
World Scientific News; 2019, 118; 100-114
2392-2192
Pojawia się w:
World Scientific News
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Novel s-Triazinyl Schiff Base/Chalcone Congeners: Rational, Synthesis, Antimicrobial and Anti-TB Evaluation
Autorzy:
Lakum, H. P.
Shah, D. R.
Chikhalia, K. H.
Powiązania:
https://bibliotekanauki.pl/articles/412603.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
antimicrobial
Anti-TB
s-Triazine
Schiff base
Chalcone
Opis:
The occurrence of Multi Drug Resistant (MDR) infectious microbial strains has been increased upto alarming level which affects the public health worldwide. To cure this problem, a library of s-triazinyl derivatives comprising schiff base or chalcone motif have been rationalized, synthesized and screened for their in vitro antibacterial activity against five bacterial strains (Staphylococcus aureus MTCC 96, Bacillus subtilis MTCC 441, Escherichia coli MTCC 739, Pseudomonas aeruginosa MTCC 741 and Klebsiella pneumoniae MTCC 109) and four fungal strains (Aspergillus niger MTCC 282, Aspergillus fumigates MTCC 343, Aspergillus clavatus MTCC 1323, Candida albicans MTCC 183) using broth dilution technique. All the newly synthesized scaffolds were further evaluated for their in vitro anti-TB efficacy against the tubercular strain (Mycobacterium tuberculosis H37Rv) using Lowenstein-Jensen MIC method. All the derivatives were well characterized by IR, 1H NMR, 13C NMR, elemental analysis as well as mass spectroscopy.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 19, 1; 56-73
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Synthesis and in vitro antimicrobial evaluation of amine substituted s-triazine based thiazolidinone/chalcone hybrids
Autorzy:
Shah, D. R.
Lakum, H. P.
Chikhalia, K. H.
Powiązania:
https://bibliotekanauki.pl/articles/412622.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
Antibacterial
Antifungal
Chalcone
s-Triazine
4-thiazolidinone
Opis:
In an attempt to control multidrug resistant dilemma, a library of s-triazine based on two novel series of thiazolidinone (4a-e) and chalcone (7a-e) derivatives were designed and synthesized with simple and efficient etiquette. The newly synthesized compounds were studied for efficacy against several bacteria (Staphylococcus Aureus, Bacillus Cereus, Pseudomonas Aeruginosa, Klebsiella Pneumoniae,) and fungi (Candida Albicans, Aspergillus Clavatus) using the broth dilution technique. Compound 7d was the best bioactive desired antibacterial analogue with less MIC value against different tested strains. Results of bioassay study revealed the future hope of the potent drug-candidate based on s-triazine scaffold. All the final synthesized compounds were characterized by IR, 1 H NMR, 13 C NMR, mass and elemental analysis.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 17, 2; 207-219
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Phase Transition in Quasi-Two-Dimensional Horizontally Driven Granular System
Autorzy:
Shah, S.
Li, Y.
Khan, W.
Din, N.
Chand, R.
Powiązania:
https://bibliotekanauki.pl/articles/1489921.pdf
Data publikacji:
2012-03
Wydawca:
Polska Akademia Nauk. Instytut Fizyki PAN
Tematy:
81.05.Rm
64.60.-i
Opis:
In an experimental setup, consisting of quasi-two-dimensional square cell, the motion of monodisperse spherical steel balls is studied. The cell is vibrated horizontally to eradicate the compaction of balls due to gravity. By raising the number density of the steel balls, the dilute fluid has been gradually alternated into dense fluid. The temperature of granular media, along the driven and transverse directions, has been found to be anisotropic. Transition from granular gas to the liquid-like fluid has been observed. The radial distribution function of the balls in the cell is investigated for the authentication of the structural changes. Furthermore, the fast Fourier transformation for the 2D system is carried out to confirm these changes.
Źródło:
Acta Physica Polonica A; 2012, 121, 3; 699-702
0587-4246
1898-794X
Pojawia się w:
Acta Physica Polonica A
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Acid-Promoted Synthesis of Imidazolyl-Pyrazole Derivatives via a Multicomponent Reaction Using Ultra Sound Irradiation
Autorzy:
Baria, B.
Viradiya, D.
Kotadiya, V.
Kakadiya, R.
Shah, A.
Powiązania:
https://bibliotekanauki.pl/articles/412490.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
Imidazole
ultrasound irradiation
Imidazolyl-Pyrazole
Benzil
Opis:
Some new imidazolyl pyrazole derivatives have been synthesized using benzil, ammonium acetate, and heterocyclic aldehyde in ethanol and acetic acid under ultra sound irradiation. The obtained products using this approach are having high purity and good in yield. By conducting the reactions in ethanol, the solid products were precipitated out and could be isolated simply by filtration. The synthesized compounds were characterized by various analytical techniques such as 1H and 13C NMR and further supported by mass spectroscopy.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 11, 3; 277-283
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Highly efficient and eco-friendly one-pot synthesis of penta substitute pyrrole derivatives under catalyst-free conditions
Autorzy:
Viradiya, D. J.
Baria, B. H.
Kakadiya, R.
Kotadiya, V. C.
Shah, A.
Powiązania:
https://bibliotekanauki.pl/articles/412605.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
one-pot synthesis
penta-substituted pyrrole derivatives
multi-component reactions
Opis:
An eco-friendly and efficient one-pot synthesis of penta-substituted pyrrole derivatives via a four-component reaction of maldrum’s acid, arylglyoxal monohydrate, dimethyl but-2-yne-dioate and amines under catalyst-free conditions in an environmentally friendly medium is described. The simple experimental procedure, catalyst-free reaction conditions, short period of conversion, and excellent yields are the advantages of the present method. Good chemical yields have been achieved without the need for chromatography and recrystallization or other purification methods.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 11, 3; 257-264
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Recent Advances in Biotechnological Methods for Wheat Gluten Immunotoxicity Abolishment – a Review
Autorzy:
Bradauskiene, Vijole
Vaiciulyte-Funk, Lina
Shah, Bakht R.
Cernauskas, Darius
Tita, Mihaela A.
Powiązania:
https://bibliotekanauki.pl/articles/1363273.pdf
Data publikacji:
2021
Wydawca:
Instytut Rozrodu Zwierząt i Badań Żywności Polskiej Akademii Nauk w Olsztynie
Tematy:
celiac disease
wheat immunogenicity
detoxified wheat
gluten hydrolysis
Opis:
Due to the increasing incidence of gluten intolerance, researchers are focusing on finding ways to eliminate immunotoxicity of wheat, this would allow the use of wheat products for gluten-intolerant consumers. The article reviews recent studies on biotechnological methods to eliminate and reduce the immunogenicity of wheat products. So far, many gluten removal methods have been proposed, but their efficacy levels were quite different. Enzymatic treatment of gluten fragments can be considered the simplest and non-invasive tool to eliminate the toxicity of gliadins and glutenins. For this purpose, various endogenous enzymes derived from cereals, and also those of bacterial, fungal, plant, and animal origin can be used in food processing. Some of the enzymes hydrolyze gluten, others block the action of toxic protein fragments. The majority of studies were carried out using lactic acid bacteria cultures, as single strains or in consortia. Satisfactory results have been achieved using bacterial and plant enzymes, but the complete elimination of gluten immunogenicity is still possible by using fungal proteases, engineered enzymes or combining several treatments, for example, by using lactic acid fermentation or germination with fungal proteases. However, the question of how degradation of gluten affects the quality of flour (dough) in practice remains unanswered. It is not clear whether the products of such wheat flour are better and safer than those made from starches and whether their price and quality are acceptable to consumers. The insights presented in this review will be helpful to other researchers and cereal-based food producers in choosing ways to reduce gluten immunogenicity.
Źródło:
Polish Journal of Food and Nutrition Sciences; 2021, 71, 1; 5-20
1230-0322
2083-6007
Pojawia się w:
Polish Journal of Food and Nutrition Sciences
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Experimental and numerical determination of apparent mass variation of granular media confined in silo geometry
Autorzy:
Qadir, Abdul
Ispalove, Nurlybek
Ali, Asim
Chand, R.
Shah, M.
Khan, Asif
Hussain, Kashif
Powiązania:
https://bibliotekanauki.pl/articles/1070521.pdf
Data publikacji:
2016-03
Wydawca:
Polska Akademia Nauk. Instytut Fizyki PAN
Tematy:
83.80.Fg
45.70.Cc
45.70.-n
Opis:
Granular materials have vast applications both in industry and in daily life. They display quite interesting and exceptional properties different from the other known forms of matter. To investigate the complex properties of particulate materials, experimental, analytical, and numerical techniques have been employed. In this paper the results of experimental and numerical tests of various grain sizes and coefficient of friction between granules and cylindrical walls on the mass measured at bottom of container, known as apparent mass, are reported. It is revealed that apparent mass augments with the grain size. Moreover, it is also found that the variation in apparent mass measurement is strongly dependent on bead diameter rather than the silo size. The results suggest that the conversion of vertical stresses into horizontal in silo is mainly due to the friction between the grain and system boundary than the arching phenomenon.
Źródło:
Acta Physica Polonica A; 2016, 129, 3; 378-382
0587-4246
1898-794X
Pojawia się w:
Acta Physica Polonica A
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Synthesis, Characterization and Biological evaluation of some newer 5-[6-chloro/fluoro/nitro-2-(p-chloro/ fluoro/ methyl phenyl)-quinolin-4-yl]-1,3,4-oxadiazole-2-thiols
Autorzy:
Faldu, V. J.
Talpara, P. K.
Bhuva, N. H.
Vachharajani, P. R.
Shah, V. H.
Powiązania:
https://bibliotekanauki.pl/articles/412197.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
Quinolines
1,3,4-oxadiazole-2-thiols
therapeutic agents
antimicrobial assai
Opis:
Recent study shows that quinolines represent one of the most active classes of compounds possesses wide spectrum biodynamic activities and use as potent therapeutic agents. In present research work, 5-[6-chloro/fluoro/nitro-2-(p-chloro/fluoro/methyl phenyl)-quinolin-4-yl]-1,3,4-oxadiazole-2-thiols have been synthesized by condensation of substituted quinoline-4-carbohydrazides and mixture of carbon disulphide and potassium hydroxide. All of these compounds were screened for their in vitroanti microbial assay against gram (+ve), gram (-ve) bacteria and fungi activity compared with standard drugs viz., Ampicilin, Chloramphenicol, Ciprofloxacin, Norfloxacin, Griseofulvin and Nystatin at different concentrations.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 6; 26-32
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Novel conversion of 4-aminoquinolines to new tricyclic (R,S)-3-methylazeto[3,2-c] quinolin-2(2aH)-ones and versatile one step synthesis of N-(quinolin-4-yl) carbamates from 4-aminoquinolines
Autorzy:
Kotadiya, V. C.
Viradiya, D. J.
Baria, B. H.
Kanzariya, J. S.
Kakadiya, R.
Shah, A.
Powiązania:
https://bibliotekanauki.pl/articles/412269.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
quinolin
carbamates
azeto-quinolinone
aminoquinolines
Opis:
Reaction of 4-aminoquinolines with 4-nitrophenyl chloroformate have resulted in finding a novel transformation of 4-aminoquinolines to tricyclic (R,S)-3-methylazeto[3,2-c]quinolin-2(2aH)-ones. The structure of azeto-quinolinone was determined via spectroscopic and chemical methods. Various alcohols were used as nucleophiles to open the 1-azetinone ring to give the corresponding N-(quinolin-4-yl)carbamates in good yields. We also found a new and versatile one step synthesis of N-(quinolin-4-yl)carbamates by reacting 4-aminoquinolines with alkyl chloroformates in the presence of anhyd K2CO3 in acetonitrile.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 11, 3; 265-276
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł

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