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Wyszukujesz frazę "Shah, H." wg kryterium: Autor


Wyświetlanie 1-28 z 28
Tytuł:
Modeling computational studies of modified drug molecules binding to the LRRK2 protein in the treatment of Parkinson’s disease
Autorzy:
Shah, H.
Darsey, J. A.
Powiązania:
https://bibliotekanauki.pl/articles/284742.pdf
Data publikacji:
2018
Wydawca:
Akademia Górniczo-Hutnicza im. Stanisława Staszica w Krakowie. Polskie Towarzystwo Biominerałów
Tematy:
LRRK2 proteins
Parkinson
Computational Modeling
IC50
Density Functional Theory
DFT
Opis:
Parkinson’s disease is a neurodegenerative and progressive disease of the central nervous system. It affects more than 10 million patients worldwide and the symptoms allow for little to no control for movement. These symptoms appear because the chemical messenger dopamine is being made in small quantities from impaired cells. However, the disease often forms when there is a mutation in the LRRK2 gene, as the functions of the protein become abnormal. The IC50 value is essential information about molecules because it measures their effectiveness. The goal of this research was to design molecules with a lower IC50 value. This was first done by modeling molecules on the molecular modeling program, Gaussian 09. Modifications were made to molecules that were said to bind to the LRRK2 protein. Modifications ranged from adding a single atom or replacing atoms with groups. After running these molecules on the program, the total energy was found. Using the equation found from the correlation between 1/IC50 and the total energy, the IC50 value was predicted for each of the modified molecules. Many of the modified molecules portrayed a positive percent difference between the original IC50 value and the new one. This saves both time and money because the molecules with lower IC50 values can be made, preserving the resources. After creating the molecule with a low IC50 value, further experimental procedures can be taken; this is a large step in assisting researchers to reach a potential treatment because it is more efficient.
Źródło:
Engineering of Biomaterials; 2018, 21, 145; 2-7
1429-7248
Pojawia się w:
Engineering of Biomaterials
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Music Playlist Generation using Facial Expression Analysis and Task Extraction
Autorzy:
Sen, A.
Popat, D.
Shah, H.
Kuwor, P.
Johri, E.
Powiązania:
https://bibliotekanauki.pl/articles/908868.pdf
Data publikacji:
2016
Wydawca:
Uniwersytet Marii Curie-Skłodowskiej. Wydawnictwo Uniwersytetu Marii Curie-Skłodowskiej
Tematy:
facial expression analysis
emotion recognition
feature extraction
viola jones face detection
gabor filter
adaboost
k-NN algorithm
task extraction
music classification
playlist generation
Opis:
In day to day stressful environment of IT Industry, there is a truancy for the appropriate relaxation time for all working professionals. To keep a person stress free, various technical or non-technical stress releasing methods are now being adopted. We can categorize the people working on computers as administrators, programmers, etc. each of whom require varied ways in order to ease themselves. The work pressure and the vexation of any kind for a person can be depicted by their emotions. Facial expressions are the key to analyze the current psychology of the person. In this paper, we discuss a user intuitive smart music player. This player will capture the facial expressions of a person working on the computer and identify the current emotion. Intuitively the music will be played for the user to relax them. The music player will take into account the foreground processes which the person is executing on the computer. Since various sort of music is available to boost one's enthusiasm, taking into consideration the tasks executed on the system by the user and the current emotions they carry, an ideal playlist of songs will be created and played for the person. The person can browse the playlist and modify it to make the system more flexible. This music player will thus allow the working professionals to stay relaxed in spite of their workloads.
Źródło:
Annales Universitatis Mariae Curie-Skłodowska. Sectio AI, Informatica; 2016, 16, 2; 1-6
1732-1360
2083-3628
Pojawia się w:
Annales Universitatis Mariae Curie-Skłodowska. Sectio AI, Informatica
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Coordinated production, ordering, shipment and pricing model for supplier-retailer inventory system under trade credit
Autorzy:
Shah, Nita H.
Naik, Monika K.
Powiązania:
https://bibliotekanauki.pl/articles/406551.pdf
Data publikacji:
2019
Wydawca:
Politechnika Wrocławska. Oficyna Wydawnicza Politechniki Wrocławskiej
Tematy:
defective item
production inventory system
supply chain of two players
time-price
credit
dependent demand
element uszkodzony
system inwentaryzacji produkcji
łańcuch dostaw
kredyt
popyt zależny
Opis:
The objective of this article is to maximize the joint profit for supplier and retailer by constructing a combined supplier–retailer inventory model wherein supplier and retailer both have implemented trade credit policies, and some defective items are received by the retailer. The customer’s demand is expressed as a function of time, price and credit period, which is appropriate for the products for which demand increases initially and after some time it starts to decrease. Production, directly proportional to the customer’s demand rate, is considered as one of the decision variables for the purpose of reducing the holding cost of the supplier. The article estimates the optimum replenishment cycle, customer’s credit period, retail selling price by a classical optimization technique. For validation of the derived model, various numerical examples are demonstrated. Finally, implementing sensitivity analysis on the decision variables by varying the inventory parameters, effective managerial insights are generated which is beneficial for the players of supply chain by practically gaining the maximum joint profit through advising to opt for the case N ≤ M ≤ T , i.e., when the customer’s trade credit period offered by the retailer is lesser than the retailer’s trade credit period offered by the supplier and which is lesser than the replenishment cycle length.
Źródło:
Operations Research and Decisions; 2019, 29, 2; 55-76
2081-8858
2391-6060
Pojawia się w:
Operations Research and Decisions
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
An efficient one-pot multicomponent synthesis and characterization of 5-cyano-1,2,3,4-tetrahydropyrimidine derivatives
Autorzy:
Vaghasiya, R. G.
Shah, V. H.
Powiązania:
https://bibliotekanauki.pl/articles/411702.pdf
Data publikacji:
2015
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
substituted pyrazole-4-carbaldehyde
5-cyano-1,2,3,4-tetrahydropyrimidine derivatives
multi component reaction
non-chromatographic method
Opis:
A series of pyrimidine-5-carbonitrile derivatives was efficiently synthesized via one-pot, multi component reaction (MCRs) of 1,3-bifunctional synthon (ethylcyano acetate), substituted pyrazole-4-carbaldehyde, and thiourea/urea in the presence of basic catalyst. The key advantages of this process are high yields, shorter reaction times, easy work-up, and purification of products by non-chromatographic method.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2015, 40; 51-60
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Inventory models and trade credit: a review
Autorzy:
Soni, H.
Shah, N. H.
Jaggi, C. K.
Powiązania:
https://bibliotekanauki.pl/articles/969900.pdf
Data publikacji:
2010
Wydawca:
Polska Akademia Nauk. Instytut Badań Systemowych PAN
Tematy:
lot-size model
trade credit
deterioration
probabilistic demand
Opis:
This article reviews the literature on quantitatively oriented approaches for determining the optimal lot-size when supplier offers credit period to the retailer to settle their account. An attempt is made to provide an up-to-date review of existing literature, concentrating on descriptions of the types of problems that have been solved and important structural results.
Źródło:
Control and Cybernetics; 2010, 39, 3; 867-882
0324-8569
Pojawia się w:
Control and Cybernetics
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Optimal credit period and ordering quantity for credit dependent trended demand and deteriorating items with maximum lifetime
Autorzy:
Shah, N. H.
Shah, D. B.
Patel, D. G.
Powiązania:
https://bibliotekanauki.pl/articles/970075.pdf
Data publikacji:
2015
Wydawca:
Polska Akademia Nauk. Instytut Badań Systemowych PAN
Tematy:
inventory
trended demand
trade credit
default risk
deterioration
maximum lifetime
Opis:
In this paper, an inventory system is analyzed regarding a trended demand. The seller offers its buyer a credit period for settling the account, which attracts more buyers and enhances market demand. However, the offer of credit period leads to default risk for the supplier. The units in inventory are deteriorating continuously and also have definite maximum lifetime. The aim is to maximize the profit of the retailer. Numerical examples are given to validate the developed mathematical model. Sensitivity analysis is performed to obtain the critical inventory parameters and deduce the managerial strategies.
Źródło:
Control and Cybernetics; 2015, 44, 2; 311-320
0324-8569
Pojawia się w:
Control and Cybernetics
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
An EOQ model with time dependent deterioration under discounted cash flow approach when supplier credits are linked to order quantity
Autorzy:
Shah, B. J.
Shah, N. H.
Shah, Y. K.
Powiązania:
https://bibliotekanauki.pl/articles/970398.pdf
Data publikacji:
2007
Wydawca:
Polska Akademia Nauk. Instytut Badań Systemowych PAN
Tematy:
time dependent deterioration
discounted cashflows (DCF) approach
supplier credit linked to order quantity
Opis:
This article deals with an inventory model under a situation in which the supplier offers the purchaser some credit period if the purchaser orders a large quantity. Shortages are not allowed. The effects of the inflation rate on purchase price, ordering price and inventory holding price, time dependent deterioration of units and permissible delay in payment are discussed. A mathematical model is developed when units in inventory are subject to time dependent deterioration under inflation when the supplier offers a permissible delay to the purchaser if the order quantity is greater than or equal to a pre-specified quantity. Optimal solution is obtained and algorithm is given to find the optimal order quantity and replenishment time, which minimizes the total cost of an inventory system in different scenarios. The paper concludes with a numerical example to illustrate the theoretical results and interdependence of parameters is studied for the optimal solutions.
Źródło:
Control and Cybernetics; 2007, 36, 2; 405-423
0324-8569
Pojawia się w:
Control and Cybernetics
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
A rapid, convient and diversified-multicomponent synthesis and characterization of pyrano[2,3-b]indoles
Autorzy:
Ghodasara, H. B.
Singala, P. M.
Shah, V. H.
Powiązania:
https://bibliotekanauki.pl/articles/412134.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
1,3-bifunctional synthon
Pyrano[2,3-b]indoles
multi component reaction
non-chromatographic metod
Opis:
A series of pyrano[2,3-b]indoles, was efficiently synthesized via one-pot, multi component reaction (MCRs) of 1,3-bifunctional synthon(malononitrile/ethylcyano acetate), aromatic aldehydes and oxiindole in the presence of various basic catalyst. The key advantages of this process are high yields, shorter reaction times, easy work-up, and purification of products by non-chromatographic method.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 7; 69-76
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Synthesis, Characterization and Biological evaluation of 6-substituted-2-(substituted-phenyl)-quinoline derivatives bearing 4-amino-1,2,4-triazole-3-thiol ring at C-4 position
Autorzy:
Vaghasiya, R. G.
Ghodasara, H. B.
Vachharajani, P. R.
Shah, V. H.
Powiązania:
https://bibliotekanauki.pl/articles/412211.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
Quinoline, 4-amino-1,2,4-triazole-3-thiol
therapeutic agents
antimicrobial assai
Opis:
Quinoline derivatives represent one of the most active classes of compounds possesses wide spectrum biodynamic activities and use as potent therapeutic agents. In this research work, a synthesis, characterization and biological evaluation of 6-substituted-2-(substituted-phenyl)-quinoline derivatives bearing 4-amino-1,2,4-triazole-3-thiol ring at C-4 position is described. The synthesis of quinoline derivatives is carried out by the reaction of substituted quinoline-4-carbohydrazides with a mixture of carbon disulphide and potassium hydroxide which further react with hydrazine hydrate to give final compounds. All of these compounds were screened for their in vitro antimicrobial assay against gram (+ve), gram (-ve) bacteria and fungi activity compared with standard drugs viz., Ampicilin, Chloramphenicol, Ciprofloxacin, Norfloxacin, Griseofulvin and Nystatin at different concentrations.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 8; 30-37
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Challenges and opportunities for the future of icampuses
Autorzy:
Thomas, A. M.
Shah, H.
Moore, P.
Evans, C.
Sharma, M.
Pham, H. V.
Osman, K.
Wilcox, A. J.
Rayson, P.
Chapman, C.
Chima, P.
Athwal, C.
While, D.
Powiązania:
https://bibliotekanauki.pl/articles/952933.pdf
Data publikacji:
2013
Wydawca:
Akademia Górniczo-Hutnicza im. Stanisława Staszica w Krakowie. Wydawnictwo AGH
Tematy:
education
icampus
sensors
context
Web 2.0
Opis:
Meeting the educational needs of students currently requires moving toward collaborative electronic and mobile learning systems that parallel the vision of Web 2.0. However, factors such as data freedom, brokerage, interconnectivity and the Internet of Things add to a vision for Web 3.0 that will require consideration in the development of future campus-based, distance and vocational study. So, education can, in future, be expected to require deeper technological connections between students and learning environments, based on significant use of sensors, mobile devices, cloud computing and rich-media visualization. Therefore, we discuss challenges associated with such a futuristic campus context, including how learning materials and environments may be enriched by it. As an additional novel element the potential for much of that enrichment to be realized through development by students, within the curriculum, is also considered. We will conclude that much of the technology required to embrace the vision of Web 3.0 in education already exists, but that further research in key areas is required for the concept to achieve its full potential.
Źródło:
Computer Science; 2013, 14 (1); 5-25
1508-2806
2300-7036
Pojawia się w:
Computer Science
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Synthesis, Characterization and Biological evaluation of some newer 5-[6-chloro/fluoro/nitro-2-(p-chloro/ fluoro/ methyl phenyl)-quinolin-4-yl]-1,3,4-oxadiazole-2-thiols
Autorzy:
Faldu, V. J.
Talpara, P. K.
Bhuva, N. H.
Vachharajani, P. R.
Shah, V. H.
Powiązania:
https://bibliotekanauki.pl/articles/412197.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
Quinolines
1,3,4-oxadiazole-2-thiols
therapeutic agents
antimicrobial assai
Opis:
Recent study shows that quinolines represent one of the most active classes of compounds possesses wide spectrum biodynamic activities and use as potent therapeutic agents. In present research work, 5-[6-chloro/fluoro/nitro-2-(p-chloro/fluoro/methyl phenyl)-quinolin-4-yl]-1,3,4-oxadiazole-2-thiols have been synthesized by condensation of substituted quinoline-4-carbohydrazides and mixture of carbon disulphide and potassium hydroxide. All of these compounds were screened for their in vitroanti microbial assay against gram (+ve), gram (-ve) bacteria and fungi activity compared with standard drugs viz., Ampicilin, Chloramphenicol, Ciprofloxacin, Norfloxacin, Griseofulvin and Nystatin at different concentrations.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 6; 26-32
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Synthesis of novel 2-mercapto-4-(p-aminophenyl sulphonylamino)-6-(aryl)-pyrimidine-5-carboxamide derivatives via the Biginelli reaction
Autorzy:
Bhuva, N. H.
Gothalia, V. K.
Singala, P. M.
Talpara, P. K.
Faldu, V. J.
Shah, V. H.
Powiązania:
https://bibliotekanauki.pl/articles/412069.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
2-mercapto-4-(p-aminophenylsulphonylamino)-6-(aryl)-pyrimidine-5-carboxamide
Biginelli condensation
Opis:
Series of 2-mercapto-4-(p-aminophenylsulphonylamino)-6-(aryl)-pyrimidine-5-carboxamide Aa-h were synthesized via the biginelli condensation. 2-mercapto-4-amino-6-(aryl)-pyrimidine-5-carboxamide react with p-acetamidophenylsulphonylchloride in the presence of pyridine 2 to form 2-mercapto-4-(p-acetamidophenylsulphonylamino)-6-(aryl)-pyrimidine-5-carboxamide 3. It was treated with diluted HCl under reflux afforded 2-mercapto-4-(p-aminophenylsulphonylamino)-6-(aryl)-pyrimidine-5-carboxamide A a-h. The newly synthesized compounds were characterized by elemental analyses, infrared (IR), 1H NMR and 13 C NMR spectroscopic investigation.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 17, 2; 168-173
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Maximizing power output of a partially shaded total-cross-tied photovoltaic array
Autorzy:
Shah, N. S.
Patel, H. H.
Powiązania:
https://bibliotekanauki.pl/articles/136262.pdf
Data publikacji:
2017
Wydawca:
EEEIC International Barbara Leonowicz Szabłowska
Tematy:
current compensation
voltage equalization
MPPT
partial shading
TCT configuration
Opis:
Non-uniform conditions on the modules of the PV array, especially, partial shading reduces the output of the PV array to a large extent. The shaded module in a string limits the current of the entire string and hence, the output power of the string. The output power under such conditions is reported to be higher for total-cross-tied (TCT) configuration. This paper describes two different approaches, one based on current compensation (current equalization) and another based on voltage equalization, to extract higher power from the partially shaded total-cross-tied photovoltaic array. The TCT configuration is considered to minimize the number of converters, sensors, cost and complexity involved. The additional converters in the two distinct approaches evaluated here operate only when the partial shading occurs and are controlled to minimize the current and voltage miss-matches. The analysis and the control algorithm are presented. Simulation results obtained in MATLAB/Simulink are included to demonstrate the effectiveness of both methods and the relative merits and demerits of these approaches are highlighted.
Źródło:
Transactions on Environment and Electrical Engineering; 2017, 2, 1; 10-18
2450-5730
Pojawia się w:
Transactions on Environment and Electrical Engineering
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Synthesis and antimicrobial screening of some new pyrimido[1,2-a]benzimidazole derivatives
Autorzy:
Shah, N. M.
Joshi, H. S.
Powiązania:
https://bibliotekanauki.pl/articles/411967.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
2-aminobenzimidazole
pyrimido[1,2-a]benzimidazole
chalcone
antimicrobial activity azoloazine
Opis:
Some new pyrimido[1,2-a]benzimidazole derivatives were synthesized by reacting 2-amino benzimidazole and chalcones in n-butanol at reflux temperature. In our present study we have used various heterocyclic chalcones derived from furfural and substituted acetophenones. All synthesized compounds were characterized by IR, 1H NMR and Mass spectroscopy. All synthesized compounds were screened for their antimicrobial activity against gram positive and gram negative bacteria which showed moderate to good activity.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 6; 56-60
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Novel s-Triazinyl Schiff Base/Chalcone Congeners: Rational, Synthesis, Antimicrobial and Anti-TB Evaluation
Autorzy:
Lakum, H. P.
Shah, D. R.
Chikhalia, K. H.
Powiązania:
https://bibliotekanauki.pl/articles/412603.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
antimicrobial
Anti-TB
s-Triazine
Schiff base
Chalcone
Opis:
The occurrence of Multi Drug Resistant (MDR) infectious microbial strains has been increased upto alarming level which affects the public health worldwide. To cure this problem, a library of s-triazinyl derivatives comprising schiff base or chalcone motif have been rationalized, synthesized and screened for their in vitro antibacterial activity against five bacterial strains (Staphylococcus aureus MTCC 96, Bacillus subtilis MTCC 441, Escherichia coli MTCC 739, Pseudomonas aeruginosa MTCC 741 and Klebsiella pneumoniae MTCC 109) and four fungal strains (Aspergillus niger MTCC 282, Aspergillus fumigates MTCC 343, Aspergillus clavatus MTCC 1323, Candida albicans MTCC 183) using broth dilution technique. All the newly synthesized scaffolds were further evaluated for their in vitro anti-TB efficacy against the tubercular strain (Mycobacterium tuberculosis H37Rv) using Lowenstein-Jensen MIC method. All the derivatives were well characterized by IR, 1H NMR, 13C NMR, elemental analysis as well as mass spectroscopy.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 19, 1; 56-73
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Synthesis and in vitro antimicrobial evaluation of amine substituted s-triazine based thiazolidinone/chalcone hybrids
Autorzy:
Shah, D. R.
Lakum, H. P.
Chikhalia, K. H.
Powiązania:
https://bibliotekanauki.pl/articles/412622.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
Antibacterial
Antifungal
Chalcone
s-Triazine
4-thiazolidinone
Opis:
In an attempt to control multidrug resistant dilemma, a library of s-triazine based on two novel series of thiazolidinone (4a-e) and chalcone (7a-e) derivatives were designed and synthesized with simple and efficient etiquette. The newly synthesized compounds were studied for efficacy against several bacteria (Staphylococcus Aureus, Bacillus Cereus, Pseudomonas Aeruginosa, Klebsiella Pneumoniae,) and fungi (Candida Albicans, Aspergillus Clavatus) using the broth dilution technique. Compound 7d was the best bioactive desired antibacterial analogue with less MIC value against different tested strains. Results of bioassay study revealed the future hope of the potent drug-candidate based on s-triazine scaffold. All the final synthesized compounds were characterized by IR, 1 H NMR, 13 C NMR, mass and elemental analysis.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 17, 2; 207-219
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Synthesis and antimicrobial activity of some new imidazolinone derivatives containing benzimidazole
Autorzy:
Mehta, P.
Davadra, P.
Shah, N.
Joshi, H.
Powiązania:
https://bibliotekanauki.pl/articles/411949.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
benzimidazole
imidazolinone
antimicrobial activity
Opis:
In this study some new o-benzimidazol-2'-yl-benzamido-p'-benzamido-2-phenyl-4-substituted phenyl-5-oxo-Imidazolines 3a-3j were synthesized. To synthesized target molecules we used various substituted oxazolone derivatives, synthesized from substituted benzaldehyde with hippuric acid. Substituted oxazolones 2a-2j were reacted with carbohydrazide derivative of benzimidazole 1 in presence of pyridine as base to obtained substituted imidazolinone derivatives. All synthesized compounds were characterized by IR, 1H NMR, elemental analysis and further supported by mass spectroscopy. All synthesized compounds were screened for their antimicrobial activity against gram positive and gram negative bacteria which showed moderate to good activity. All compounds showing good to moderate active against fungal strain as compare to standard drug.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 10; 74-80
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Synthesis and characterization of some new Schiff bases of 2-oxonaphtho[2,1-b][1,4]oxazine
Autorzy:
Chovatiya, P.
Mehta, C.
Senjani, H.
Shah, A.
Joshi, H. S.
Powiązania:
https://bibliotekanauki.pl/articles/411737.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
2-Oxonaphtho[2,1-b][1,4]oxazine
Schiff base
Opis:
The literature review reveal that [1,4]-oxazine derivatives represent one of the most active classes of compounds possessing wide spectrum of biodynamic activities and use as potent therapeutic agents. In the present work, a series of Schiff base of 2-(2,3-dihydro-2-oxonaphtho[2,1-b][1,4]oxazin-1-yl)acetohydrazide, 5a-5j has been synthesized using 1-aminonaphthalen-2-ol. Various aromatic aldehyde were react with carbohydrazide 4 in the presence of acid to produce the 2-oxonaphtho[2,1-b][1,4]oxazin Schiff base derivatives with good yields. All synthesized compounds were characterized by IR, NMR and Mass spectrometry analysis.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 12; 26-30
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Synthesis, characterization of biologically potent novel chalcones bearing urea, thiourea and acetamide linkages
Autorzy:
Mewada, N. S.
Shah, D. R.
Chikhalia, K. H.
Powiązania:
https://bibliotekanauki.pl/articles/412032.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
Chalcone
urea
thiourea
acetamide
antimicrobial activity and antifungal activity
Opis:
Three series of some novel chalcone based urea, thiourea and acetamide derivatives were designed, synthesized and screened for their antimicrobial and antifungal activities. All the synthesized compounds are first reported. The structures of the compounds were elucidated with the aid of elemental analysis and spectral methods including IR, 1H-NMR spectral data. The prepared compounds were evaluated for antibacterial activity against two Gram-positive bacteria (Staphylococcus aureus, Staphylococcus pyogenus), two Gram-negative bacteria (Pseudomonas aeruginosa, Escherichia coli). The title compounds were also investigated for their antifungal activity using the broth micro dilution method. The bioassay results showed that compounds a few compounds showed good to superior in vitro antibacterial and antifungal activity.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 17, 3; 281-294
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Disparity of a Seat Cushion and Its Influence on Postural Control
Autorzy:
Nag, P.K.
Nag, A.
Vyas, H.
Shah, P.
Powiązania:
https://bibliotekanauki.pl/articles/89723.pdf
Data publikacji:
2013
Wydawca:
Centralny Instytut Ochrony Pracy
Tematy:
cushion
foam
cotton
centre of pressure measurements
postural control
kontrola postawy ciała
postawa ciała
siedzenie
kontrola równowagi
Opis:
Properties of supporting surfaces of a seat have an influence on postural control. Centre of pressure (COP) displacement parameters reflect both the balance controlling process and movements of the centre of a mass of entire body. The subjects of the study were 9 healthy men. A seat cushion was examined with a 2-force platform setup. Force exertion at a seat pan and feet and COP displacement at a seat pan were measured to analyse postural control. Analysis of variance determined the differences in postural control depending on a cushion type among the subjects. Significant differences in COP displacement parameters were in COP trajectory length, medio-lateral COP displacement and COP velocity. The results of the study showed that foam cushion ensures better postural control.
Źródło:
International Journal of Occupational Safety and Ergonomics; 2013, 19, 4; 573-581
1080-3548
Pojawia się w:
International Journal of Occupational Safety and Ergonomics
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Synthesis, characterization and docking studies of some novel xanthene derivatives
Autorzy:
Bhatt, Aditya H.
Shah, Viral R.
Rawal, Rakesh M.
Powiązania:
https://bibliotekanauki.pl/articles/1075739.pdf
Data publikacji:
2019
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
Antimicrobial activity
Docking studies
Hantzsch synthesis
Xanthene
Opis:
The synthesis of a novel xanthene derivatives bearing dimedone as an excellent precursor has been achieved by applying one pot three component Hantzsch type condensation. The newly synthesized compounds were characterized by spectral and elemental analyses. All synthesized compounds undergo docking studies and biological screening for antimicrobial activity against Gram-positive bacteria, Gram-negative bacteria and fungal species. Among all the tested compounds, it was found that compound 3c, 3d, 3g and 3h revealed better activities against the Gram-positive rather than the Gram-negative bacteria whereas results of docking studies revealed that compounds 3b, 3g and 3i showed best binding affinity towards ATP binding pocket of Human PIM1 kinase receptor through steric favorable and H-bond interactions.
Źródło:
World Scientific News; 2019, 118; 100-114
2392-2192
Pojawia się w:
World Scientific News
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Assessment of Eco-Friendly Natural Antimicrobial Textile Finish Extracted from Aloe Vera and Neem Plants
Ocena ekologicznych naturalnych preparacji antymikrobowych tekstyliów uzyskanych z udziałem ekstraktów z aloesu i miodli indyjskiej
Autorzy:
Khurshid, M. F.
Ayyoob, M.
Asad, M.
Shah, S. N. H.
Powiązania:
https://bibliotekanauki.pl/articles/233713.pdf
Data publikacji:
2015
Wydawca:
Sieć Badawcza Łukasiewicz - Instytut Biopolimerów i Włókien Chemicznych
Tematy:
eco-friendly
antimicrobial
natural textile finish
aloe vera extraction
neem extraction
ekologiczne preparacje
przeciwbakteryjne preparacje
naturalne wykończenie tkaniny
ekstrakcja z aloesu
ekstrakcja z miodli indyjskiej
Opis:
The aim of the present work was to assess an eco friendly natural antimicrobial textile finish extracted from Aloe gel and Neem plants. Extracted Aloe gel and active substance of Neem were mixed in a mordant to form a finish. Bleached cotton samples were treated with 5, 7, and 10% concentrations of Aloe gel and Neem separately. The same samples were then treated with a hybrid combination of Aloe gel and Neem (HCAN) extracts having 5, 7 and 10% concentrations. These finished samples were subjected to an antibacterial activity test against E. coli and S. aureus, an antifungal activity test against Aspergillus Niger, and a test of their durability of antibacterial finish fastness to washing by standard test methods. It was found that the hybrid combination of Aloe gel and Neem (HCAN) was an effective antibacterial and antifungal agent as compared to Aloe gel and Neem separately. It also showed good durability to washing.
Ekstrakty z żelu aloesowego i aktywnych substancji miodli indyjskiej mieszano w zaprawie barwiarskiej dla uzyskania gotowej preparacji. Bielone bawełniane próbki nasycano roztworem o stężeniu 5%, 7% i 10% żelu aloesowego i miodli indyjskiej. Te same próbki były następnie nasycane preparacją hybrydową zawierającą obydwa składniki o tym samym stężeniu. Uzyskane próbki poddano badaniom antybakteryjnym przeprowadzając testy przeciwko E. coli i S. aureus, i antygrzybicznej aktywności przeciwko Aspergillus niger. Niezależnie od tego przeprowadzano próby trwałości preparacji antybakteryjnych po praniu w standardowych warunkach. Stwierdzono, że preparacja hybrydowa obydwu składników była aktywniejsza zarówno w stosunku do bakterii i grzybów niż preparacje z użyciem jednego tylko składnika.
Źródło:
Fibres & Textiles in Eastern Europe; 2015, 6 (114); 120-123
1230-3666
2300-7354
Pojawia się w:
Fibres & Textiles in Eastern Europe
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Highly efficient and eco-friendly one-pot synthesis of penta substitute pyrrole derivatives under catalyst-free conditions
Autorzy:
Viradiya, D. J.
Baria, B. H.
Kakadiya, R.
Kotadiya, V. C.
Shah, A.
Powiązania:
https://bibliotekanauki.pl/articles/412605.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
one-pot synthesis
penta-substituted pyrrole derivatives
multi-component reactions
Opis:
An eco-friendly and efficient one-pot synthesis of penta-substituted pyrrole derivatives via a four-component reaction of maldrum’s acid, arylglyoxal monohydrate, dimethyl but-2-yne-dioate and amines under catalyst-free conditions in an environmentally friendly medium is described. The simple experimental procedure, catalyst-free reaction conditions, short period of conversion, and excellent yields are the advantages of the present method. Good chemical yields have been achieved without the need for chromatography and recrystallization or other purification methods.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 11, 3; 257-264
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Korean WA-DGNSS User Segment Software Design
Autorzy:
Shah, S. T.
Choi, W.S.
Han, W.Y.
Yun, H.
Kee, C.
Powiązania:
https://bibliotekanauki.pl/articles/116066.pdf
Data publikacji:
2013
Wydawca:
Uniwersytet Morski w Gdyni. Wydział Nawigacyjny
Tematy:
global navigation satellite system (GNSS)
Global Positioning System GPS
User Segment
GPS Data Processing Classes
Opis:
Korean WA‐DGNSS is a large scale research project funded by Ministry of Land, Transport and Maritime Affairs Korea. It aims to augment the Global Navigation Satellite System by broadcasting additional signals from geostationary satellites and providing differential correction messages and integrity data for the GNSS satellites. The project is being carried out by a consortium of universities and research institutes. The research team at Electronics and Telecommunications Research Institute is involved in design and development of data processing softwares for wide area reference station and user segment. This paper focuses on user segment software design. Korean WA‐DGNSS user segment software is designed to perform several functions such as calculation of pseudorange, ionosphere and troposphere delays, application of fast and slow correction messages, and data verification. It is based on a layered architecture that provides a model to develop flexible and reusable software and is divided into several independent, interchangeable and reusable components to reduce complexity and maintenance cost. The current version is designed to collect and process GPS and WADGNSS data however it is flexible to accommodate future GNSS systems such as GLONASS and Galileo.
Źródło:
TransNav : International Journal on Marine Navigation and Safety of Sea Transportation; 2013, 7, 1; 69-74
2083-6473
2083-6481
Pojawia się w:
TransNav : International Journal on Marine Navigation and Safety of Sea Transportation
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Novel synthesis of 3-(((E)-benzylidene)amino)-5-((Z)-3,4-dimethoxybenzylidene)-2-phenyl-3,5-dihydro-4H-imidazol-4-one derivatives as potent antimicrobial agents
Autorzy:
Manawar, Rohit B.
Parmar, Mukesh B.
Nayaka, Indresh J.
Pandit, Brinda H.
Shah, Manish K.
Powiązania:
https://bibliotekanauki.pl/articles/1066261.pdf
Data publikacji:
2019
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
4H-imidazol-4-one
A. niger
Anti-fungal
Anti-microbial Agent
Bioactivity
C. albicans
E. coli
Elemental analysis
IR spectroscopy
Mass spectroscopy
NMR spectroscopy
P. aeruginosa
S. aureus
S. pyogenes
Opis:
Novel synthesis of 4H-imidazol-4-one derivative by reaction of (Z)-3-amino-5-(3,4 dimethoxybenzylidene)-2-phenyl-3,5-dihydro-4H-imidazol-4-one with derivative of different aromatic aldehydes and Salicyldehyde. New synthesized compound are thermally stable and neither air-nor moisture sensitive at RT. Successive library of synthesized compound characterized using IR, NMR, Elemental, Mass, and its antimicrobial activity study.
Źródło:
World Scientific News; 2019, 130; 42-70
2392-2192
Pojawia się w:
World Scientific News
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Novel conversion of 4-aminoquinolines to new tricyclic (R,S)-3-methylazeto[3,2-c] quinolin-2(2aH)-ones and versatile one step synthesis of N-(quinolin-4-yl) carbamates from 4-aminoquinolines
Autorzy:
Kotadiya, V. C.
Viradiya, D. J.
Baria, B. H.
Kanzariya, J. S.
Kakadiya, R.
Shah, A.
Powiązania:
https://bibliotekanauki.pl/articles/412269.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
quinolin
carbamates
azeto-quinolinone
aminoquinolines
Opis:
Reaction of 4-aminoquinolines with 4-nitrophenyl chloroformate have resulted in finding a novel transformation of 4-aminoquinolines to tricyclic (R,S)-3-methylazeto[3,2-c]quinolin-2(2aH)-ones. The structure of azeto-quinolinone was determined via spectroscopic and chemical methods. Various alcohols were used as nucleophiles to open the 1-azetinone ring to give the corresponding N-(quinolin-4-yl)carbamates in good yields. We also found a new and versatile one step synthesis of N-(quinolin-4-yl)carbamates by reacting 4-aminoquinolines with alkyl chloroformates in the presence of anhyd K2CO3 in acetonitrile.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 11, 3; 265-276
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Equilibrium, kinetics and thermodynamic study of the adsorptive removal of methylene blue from industrial wastewater by white cedar sawdust
Autorzy:
Gardazi, Syed Mubashar H.
Shah, Jehanzeb Ali
Ashfaq, Tayyab
Sherazi, Tauqir A.
Ali, Muhammad Arif
Pervez, Arshid
Rashid, Naim
Iqbal, Javed
Amin, Bilal Ahmad Zafar
Bilal, Muhammad
Powiązania:
https://bibliotekanauki.pl/articles/207373.pdf
Data publikacji:
2019
Wydawca:
Politechnika Wrocławska. Oficyna Wydawnicza Politechniki Wrocławskiej
Tematy:
methylene blue
industrial wastewater
white cedar sawdust
WCS
dye adsorption
błękit metylenowy
ścieki przemysłowe
trociny białego cedru
adsorpcja barwników
Opis:
The study evaluated the adsorption potential of white cedar sawdust (WCS) for dye removal. WCS was chosen from five preferred, abundant waste biomasses from Pakistan. Various parameters such as contact time, adsorbent dose, dye concentration, pH, and particle size were optimized for methylene blue (MB) dye adsorption. The adsorbent was characterized by FTIR, SEM, EDX and BET analyses. The surface area of the adsorbent was 1.43 m2·g-1 and pore volume was 0.000687 cm3·g-1. The adsorption data best fitted the isotherm models of Langmuir, Temkin, Dubinin–Radushkevich, and Freundlich. The maximum experimental adsorption capacity obtained was 55.15 mg·g-1, which was in close agreement to the calculated adsorption capacity. Fitness of the pseudo-second order kinetics suggested chemisorption as the rate-limiting step. Thermodynamic study for adsorption was carried out to evaluate the Gibbs free energy (ΔG°), enthalpy (ΔH°) and entropy (ΔS°). The negative values ΔG° at the examined temperature range confirmed the spontaneous adsorption of MB onto WCS.
Źródło:
Environment Protection Engineering; 2019, 45, 3; 5-22
0324-8828
Pojawia się w:
Environment Protection Engineering
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Software Startups – A Research Agenda
Autorzy:
Unterkalmsteiner, M.
Abrahamsson, P.
Wang, X. F.
Nguyen-Duc, A.
Shah, S.
Bajwa, S. S.
Baltes, G. H.
Conboy, K.
Cullina, E.
Dennehy, D.
Edison, H.
Fernandez-Sanchez, C
Garbajosa, J.
Gorschek, T.
Klotins, E.
Hokkanen, L.
Kon, F.
Lunesu, I.
Marchesi, M.
Morgan, L.
Oivo, M.
Selig, C.
Seppänen, P.
Sweetman, R.
Tyrväinen, P.
Ungerer, C.
Yagüe, A.
Powiązania:
https://bibliotekanauki.pl/articles/953060.pdf
Data publikacji:
2016
Wydawca:
Politechnika Wrocławska. Oficyna Wydawnicza Politechniki Wrocławskiej
Tematy:
software startup
research agenda
software-intensive systems
Opis:
Software startup companies develop innovative, software-intensive products within limited time frames and with few resources, searching for sustainable and scalable business models. Software startups are quite distinct from traditional mature software companies, but also from micro-, small-, and medium-sized enterprises, introducing new challenges relevant for software engineering research. This paper’s research agenda focuses on software engineering in startups, identifying, in particular, 70+ research questions in the areas of supporting startup engineering activities, startup evolution models and patterns, ecosystems and innovation hubs, human aspects in software startups, applying startup concepts in non-startup environments, and methodologies and theories for startup research. We connect and motivate this research agenda with past studies in software startup research, while pointing out possible future directions. While all authors of this research agenda have their main background in Software Engineering or Computer Science, their interestin software startups broadens the perspective to the challenges, but also to the opportunities that emerge from multi-disciplinary research. Our audience is therefore primarily software engineering researchers, even though we aim at stimulating collaborations and research that crosses disciplinary boundaries. We believe that with this research agenda we cover a wide spectrum of the software startup industry current needs.
Źródło:
e-Informatica Software Engineering Journal; 2016, 10, 1; 89-123
1897-7979
Pojawia się w:
e-Informatica Software Engineering Journal
Dostawca treści:
Biblioteka Nauki
Artykuł
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