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Wyszukujesz frazę "Shah, D. R." wg kryterium: Autor


Wyświetlanie 1-8 z 8
Tytuł:
Synthesis, characterization of biologically potent novel chalcones bearing urea, thiourea and acetamide linkages
Autorzy:
Mewada, N. S.
Shah, D. R.
Chikhalia, K. H.
Powiązania:
https://bibliotekanauki.pl/articles/412032.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
Chalcone
urea
thiourea
acetamide
antimicrobial activity and antifungal activity
Opis:
Three series of some novel chalcone based urea, thiourea and acetamide derivatives were designed, synthesized and screened for their antimicrobial and antifungal activities. All the synthesized compounds are first reported. The structures of the compounds were elucidated with the aid of elemental analysis and spectral methods including IR, 1H-NMR spectral data. The prepared compounds were evaluated for antibacterial activity against two Gram-positive bacteria (Staphylococcus aureus, Staphylococcus pyogenus), two Gram-negative bacteria (Pseudomonas aeruginosa, Escherichia coli). The title compounds were also investigated for their antifungal activity using the broth micro dilution method. The bioassay results showed that compounds a few compounds showed good to superior in vitro antibacterial and antifungal activity.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 17, 3; 281-294
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Novel s-Triazinyl Schiff Base/Chalcone Congeners: Rational, Synthesis, Antimicrobial and Anti-TB Evaluation
Autorzy:
Lakum, H. P.
Shah, D. R.
Chikhalia, K. H.
Powiązania:
https://bibliotekanauki.pl/articles/412603.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
antimicrobial
Anti-TB
s-Triazine
Schiff base
Chalcone
Opis:
The occurrence of Multi Drug Resistant (MDR) infectious microbial strains has been increased upto alarming level which affects the public health worldwide. To cure this problem, a library of s-triazinyl derivatives comprising schiff base or chalcone motif have been rationalized, synthesized and screened for their in vitro antibacterial activity against five bacterial strains (Staphylococcus aureus MTCC 96, Bacillus subtilis MTCC 441, Escherichia coli MTCC 739, Pseudomonas aeruginosa MTCC 741 and Klebsiella pneumoniae MTCC 109) and four fungal strains (Aspergillus niger MTCC 282, Aspergillus fumigates MTCC 343, Aspergillus clavatus MTCC 1323, Candida albicans MTCC 183) using broth dilution technique. All the newly synthesized scaffolds were further evaluated for their in vitro anti-TB efficacy against the tubercular strain (Mycobacterium tuberculosis H37Rv) using Lowenstein-Jensen MIC method. All the derivatives were well characterized by IR, 1H NMR, 13C NMR, elemental analysis as well as mass spectroscopy.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 19, 1; 56-73
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Synthesis and in vitro antimicrobial evaluation of amine substituted s-triazine based thiazolidinone/chalcone hybrids
Autorzy:
Shah, D. R.
Lakum, H. P.
Chikhalia, K. H.
Powiązania:
https://bibliotekanauki.pl/articles/412622.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
Antibacterial
Antifungal
Chalcone
s-Triazine
4-thiazolidinone
Opis:
In an attempt to control multidrug resistant dilemma, a library of s-triazine based on two novel series of thiazolidinone (4a-e) and chalcone (7a-e) derivatives were designed and synthesized with simple and efficient etiquette. The newly synthesized compounds were studied for efficacy against several bacteria (Staphylococcus Aureus, Bacillus Cereus, Pseudomonas Aeruginosa, Klebsiella Pneumoniae,) and fungi (Candida Albicans, Aspergillus Clavatus) using the broth dilution technique. Compound 7d was the best bioactive desired antibacterial analogue with less MIC value against different tested strains. Results of bioassay study revealed the future hope of the potent drug-candidate based on s-triazine scaffold. All the final synthesized compounds were characterized by IR, 1 H NMR, 13 C NMR, mass and elemental analysis.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 17, 2; 207-219
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Acid-Promoted Synthesis of Imidazolyl-Pyrazole Derivatives via a Multicomponent Reaction Using Ultra Sound Irradiation
Autorzy:
Baria, B.
Viradiya, D.
Kotadiya, V.
Kakadiya, R.
Shah, A.
Powiązania:
https://bibliotekanauki.pl/articles/412490.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
Imidazole
ultrasound irradiation
Imidazolyl-Pyrazole
Benzil
Opis:
Some new imidazolyl pyrazole derivatives have been synthesized using benzil, ammonium acetate, and heterocyclic aldehyde in ethanol and acetic acid under ultra sound irradiation. The obtained products using this approach are having high purity and good in yield. By conducting the reactions in ethanol, the solid products were precipitated out and could be isolated simply by filtration. The synthesized compounds were characterized by various analytical techniques such as 1H and 13C NMR and further supported by mass spectroscopy.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 11, 3; 277-283
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Highly efficient and eco-friendly one-pot synthesis of penta substitute pyrrole derivatives under catalyst-free conditions
Autorzy:
Viradiya, D. J.
Baria, B. H.
Kakadiya, R.
Kotadiya, V. C.
Shah, A.
Powiązania:
https://bibliotekanauki.pl/articles/412605.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
one-pot synthesis
penta-substituted pyrrole derivatives
multi-component reactions
Opis:
An eco-friendly and efficient one-pot synthesis of penta-substituted pyrrole derivatives via a four-component reaction of maldrum’s acid, arylglyoxal monohydrate, dimethyl but-2-yne-dioate and amines under catalyst-free conditions in an environmentally friendly medium is described. The simple experimental procedure, catalyst-free reaction conditions, short period of conversion, and excellent yields are the advantages of the present method. Good chemical yields have been achieved without the need for chromatography and recrystallization or other purification methods.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 11, 3; 257-264
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
A new mechanism for data visualization with TSK-type preprocessed collaborative fuzzy rule based system
Autorzy:
Prasad, M.
Liu, Y.-T.
Li, D.-L.
Lin, C. -T.
Shah, R. R.
Kaiwartya, O. P.
Powiązania:
https://bibliotekanauki.pl/articles/91743.pdf
Data publikacji:
2017
Wydawca:
Społeczna Akademia Nauk w Łodzi. Polskie Towarzystwo Sieci Neuronowych
Tematy:
fuzzy interference system
collaborative clustering
fuzzy logic
big data
data visualization
Opis:
A novel data knowledge representation with the combination of structure learning ability of preprocessed collaborative fuzzy clustering and fuzzy expert knowledge of TakagiSugeno-Kang type model is presented in this paper. The proposed method divides a huge dataset into two or more subsets of dataset. The subsets of dataset interact with each other through a collaborative mechanism in order to find some similar properties within eachother. The proposed method is useful in dealing with big data issues since it divides a huge dataset into subsets of dataset and finds common features among the subsets. The salient feature of the proposed method is that it uses a small subset of dataset and some common features instead of using the entire dataset and all the features. Before interactions among subsets of the dataset, the proposed method applies a mapping technique for granules of data and centroid of clusters. The proposed method uses information of only half or less/more than the half of the data patterns for the training process, and it provides an accurate and robust model, whereas the other existing methods use the entire information of the data patterns. Simulation results show the proposed method performs better than existing methods on some benchmark problems.
Źródło:
Journal of Artificial Intelligence and Soft Computing Research; 2017, 7, 1; 33-46
2083-2567
2449-6499
Pojawia się w:
Journal of Artificial Intelligence and Soft Computing Research
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Novel conversion of 4-aminoquinolines to new tricyclic (R,S)-3-methylazeto[3,2-c] quinolin-2(2aH)-ones and versatile one step synthesis of N-(quinolin-4-yl) carbamates from 4-aminoquinolines
Autorzy:
Kotadiya, V. C.
Viradiya, D. J.
Baria, B. H.
Kanzariya, J. S.
Kakadiya, R.
Shah, A.
Powiązania:
https://bibliotekanauki.pl/articles/412269.pdf
Data publikacji:
2014
Wydawca:
Przedsiębiorstwo Wydawnictw Naukowych Darwin / Scientific Publishing House DARWIN
Tematy:
quinolin
carbamates
azeto-quinolinone
aminoquinolines
Opis:
Reaction of 4-aminoquinolines with 4-nitrophenyl chloroformate have resulted in finding a novel transformation of 4-aminoquinolines to tricyclic (R,S)-3-methylazeto[3,2-c]quinolin-2(2aH)-ones. The structure of azeto-quinolinone was determined via spectroscopic and chemical methods. Various alcohols were used as nucleophiles to open the 1-azetinone ring to give the corresponding N-(quinolin-4-yl)carbamates in good yields. We also found a new and versatile one step synthesis of N-(quinolin-4-yl)carbamates by reacting 4-aminoquinolines with alkyl chloroformates in the presence of anhyd K2CO3 in acetonitrile.
Źródło:
International Letters of Chemistry, Physics and Astronomy; 2014, 11, 3; 265-276
2299-3843
Pojawia się w:
International Letters of Chemistry, Physics and Astronomy
Dostawca treści:
Biblioteka Nauki
Artykuł
Tytuł:
Software Startups – A Research Agenda
Autorzy:
Unterkalmsteiner, M.
Abrahamsson, P.
Wang, X. F.
Nguyen-Duc, A.
Shah, S.
Bajwa, S. S.
Baltes, G. H.
Conboy, K.
Cullina, E.
Dennehy, D.
Edison, H.
Fernandez-Sanchez, C
Garbajosa, J.
Gorschek, T.
Klotins, E.
Hokkanen, L.
Kon, F.
Lunesu, I.
Marchesi, M.
Morgan, L.
Oivo, M.
Selig, C.
Seppänen, P.
Sweetman, R.
Tyrväinen, P.
Ungerer, C.
Yagüe, A.
Powiązania:
https://bibliotekanauki.pl/articles/953060.pdf
Data publikacji:
2016
Wydawca:
Politechnika Wrocławska. Oficyna Wydawnicza Politechniki Wrocławskiej
Tematy:
software startup
research agenda
software-intensive systems
Opis:
Software startup companies develop innovative, software-intensive products within limited time frames and with few resources, searching for sustainable and scalable business models. Software startups are quite distinct from traditional mature software companies, but also from micro-, small-, and medium-sized enterprises, introducing new challenges relevant for software engineering research. This paper’s research agenda focuses on software engineering in startups, identifying, in particular, 70+ research questions in the areas of supporting startup engineering activities, startup evolution models and patterns, ecosystems and innovation hubs, human aspects in software startups, applying startup concepts in non-startup environments, and methodologies and theories for startup research. We connect and motivate this research agenda with past studies in software startup research, while pointing out possible future directions. While all authors of this research agenda have their main background in Software Engineering or Computer Science, their interestin software startups broadens the perspective to the challenges, but also to the opportunities that emerge from multi-disciplinary research. Our audience is therefore primarily software engineering researchers, even though we aim at stimulating collaborations and research that crosses disciplinary boundaries. We believe that with this research agenda we cover a wide spectrum of the software startup industry current needs.
Źródło:
e-Informatica Software Engineering Journal; 2016, 10, 1; 89-123
1897-7979
Pojawia się w:
e-Informatica Software Engineering Journal
Dostawca treści:
Biblioteka Nauki
Artykuł
    Wyświetlanie 1-8 z 8

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